{"id":101598,"date":"2021-12-19T12:19:02","date_gmt":"2021-12-19T11:19:02","guid":{"rendered":"https:\/\/radioljubuski.ba\/?p=101598"},"modified":"2021-12-19T12:19:04","modified_gmt":"2021-12-19T11:19:04","slug":"martin-kondza-najmladi-doktor-znanosti-iz-gruda-i-sokovi-mogu-povecati-koncentraciju-lijeka-u-krvi","status":"publish","type":"post","link":"https:\/\/radioljubuski.ba\/index.php\/2021\/12\/19\/martin-kondza-najmladi-doktor-znanosti-iz-gruda-i-sokovi-mogu-povecati-koncentraciju-lijeka-u-krvi\/","title":{"rendered":"Martin Kond\u017ea, najmla\u0111i doktor znanosti iz Gruda: I sokovi mogu pove\u0107ati koncentraciju lijeka u krvi"},"content":{"rendered":"\n<p class=\"wp-block-paragraph\">Martin Kond\u017ea, najmla\u0111i doktor znanosti iz Gruda, s 28 godina obranio je svoj rad na Farmaceutsko-biokemijskom fakultetu Sveu\u010dili\u0161ta u Zagrebu. Nedavno je odr\u017eana i sve\u010dana promocija rada koji je nosio naziv &#8220;Mehanizam inhibicijskog u\u010dinka flavonoida na citokrom P450 3A4&#8221;, pi\u0161e Ve\u010dernji list BiH.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\"><strong>Va\u017eni enzimi<\/strong><\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Uspje\u0161ni mladi \u010dovjek zaslu\u017ean za uspostavljanje prvog nacionalnog sustava za nuspojave u BiH i zaposlenik Farmaceutskog fakulteta Sveu\u010dili\u0161ta u Mostaru govorio je za Ve\u010dernji list o svom doktorskom radu.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">&#8211; Doktorska disertacija bavila se va\u017enim enzimima u ljudskom tijelu \u2013 CYP3A4 enzimima. Ovi enzimi izme\u0111u ostaloga se nalaze u jetri, a odgovorni su za metabolizam razli\u010ditih spojeva koji ulaze u ljudski organizam (tzv. ksenobiotika), pri \u010demu kataliziraju oksidativne biotransformacije lipofilnih supstrata u polarnije metabolite, kako bi se \u0161to jednostavnije izlu\u010dili iz organizma. Budu\u0107i da na\u0161e tijelo i lijekove koje koristimo prepoznaje kao ksenobiotike, ovi enzimi odgovorni su i za metabolizam lijekova. \u0160tovi\u0161e, ovi enzimi metaboliziraju najve\u0107i broj lijekova. Razli\u010diti spojevi mogu pove\u0107avati (inducirati) aktivnost CYP3A4 enzima ili ju smanjivati (inhibirati).<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Neki od spojeva koji mogu inhibirati aktivnost CYP3A4 enzima su flavonoidi \u2013 spojevi koji se nalaze u biljkama i sastavni su dio prehrane ljudi.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Ako \u010dovjek koristi odre\u0111ene lijekove koji se metaboliziraju preko CYP3A4 enzima i primjenjuje neke flavonoide koji taj enzim mogu inhibirati, mo\u017ee do\u0107i do klini\u010dki zna\u010dajnih interakcija i do pove\u0107anih koncentracija lijeka u krvi. Iz tog razloga se, primjerice, ne preporu\u010duje piti sok od grejpfruta uz istovremeno kori\u0161tenje nekih lijekova za smanjenje masno\u0107e u krvi, za lije\u010denje visokog tlaka ili bolesti srca, lijekova protiv zgru\u0161avanja krvi i drugih lijekova &#8211; obja\u0161njava nam Kond\u017ea. Brojna su otkri\u0107a u njegovom znanstvenom radu.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\"><strong>Tra\u017eiti savjet<\/strong><\/p>\n\n\n\n<p class=\"wp-block-paragraph\">&#8211; U ovoj disertaciji otkrili smo \u010detiri nova flavonoida koja zna\u010dajno mogu inhibirati aktivnost CYP3A4 enzima \u2013 akacetin, apigenin, krizin i pinocembrin. Osim toga, opisali smo i kineti\u010dke parametre i mehanizam same inhibicije na molekularnoj razini. Takvi rezultati omogu\u0107ili su nam objavu znanstvenih radova u \u010dasopisima s visokim \u010dimbenikom odjeka, kao \u0161to je Molecules.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Iako se ova \u010detiri flavonoida u visokim koncentracijama mogu prona\u0107i u per\u0161inu, \u0161pinatu, medu i sli\u010dnoj hrani, to ne zna\u010di da \u0107e osoba s takvom prehranom imati interakciju s lijekovima. No, upravo zbog toga va\u017eno je da se ljudi prije primjene bilo kakve terapije posavjetuju s lije\u010dnicima i ljekarnicima &#8211; kazao je za Ve\u010dernji list.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Kond\u017ea je jo\u0161 jedan uspje\u0161an mladi \u010dovjek kojeg je dala Hercegovina, a on je oti\u0161ao i korak dalje s obzirom na to da je prije 30. godine ostvario brojne uspjehe te svojim otkri\u0107ima dao smjernice kako lije\u010diti ljude u budu\u0107nosti i preventivno djelovati.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Pitali smo ga i u \u010demu je tajna da ovako malo podru\u010dje daje uspje\u0161ne ljude u brojnim sferama, a koji se svojim radom isti\u010du u cijelome svijetu. &#8211; Ljudi su na ovom podru\u010dju generacijama te\u0161ko \u017eivjeli i nau\u010dili su od ni\u010dega napraviti ne\u0161to. Vjerojatno se ta genetska karakteristika prenosila s koljena na koljeno. Oskudica je tjerala ljude da razmi\u0161ljaju izvan okvira i pronalaze nove na\u010dine za rje\u0161avanje problema.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Velik utjecaj ima i zajedni\u0161tvo. Svijet se sve vi\u0161e otu\u0111uje, me\u0111utim, na\u0161i ljudi se uvijek dr\u017ee zajedno. Kako u Hercegovini, tako i u svijetu &#8211; zaklju\u010dio je Kond\u017ea.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Izvor:Vecernji.ba<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Martin Kond\u017ea, najmla\u0111i doktor znanosti iz Gruda, s 28 godina obranio je svoj rad na Farmaceutsko-biokemijskom fakultetu Sveu\u010dili\u0161ta u Zagrebu. Nedavno je odr\u017eana i sve\u010dana promocija rada koji je nosio naziv &#8220;Mehanizam inhibicijskog u\u010dinka flavonoida na citokrom P450 3A4&#8221;, pi\u0161e Ve\u010dernji list BiH. Va\u017eni enzimi Uspje\u0161ni mladi \u010dovjek zaslu\u017ean za uspostavljanje prvog nacionalnog sustava za [&hellip;]<\/p>\n","protected":false},"author":2,"featured_media":101599,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"h5ap_radio_sources":[],"footnotes":""},"categories":[1],"tags":[],"class_list":["post-101598","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-bihiregija"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.6 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Martin Kond\u017ea, najmla\u0111i doktor znanosti iz Gruda: I sokovi mogu pove\u0107ati koncentraciju lijeka u krvi - RADIO LJUBU\u0160KI<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/radioljubuski.ba\/index.php\/2021\/12\/19\/martin-kondza-najmladi-doktor-znanosti-iz-gruda-i-sokovi-mogu-povecati-koncentraciju-lijeka-u-krvi\/\" \/>\n<meta property=\"og:locale\" content=\"hr_HR\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Martin Kond\u017ea, najmla\u0111i doktor znanosti iz Gruda: I sokovi mogu pove\u0107ati koncentraciju lijeka u krvi - RADIO LJUBU\u0160KI\" \/>\n<meta property=\"og:description\" content=\"Martin Kond\u017ea, najmla\u0111i doktor znanosti iz Gruda, s 28 godina obranio je svoj rad na Farmaceutsko-biokemijskom fakultetu Sveu\u010dili\u0161ta u Zagrebu. Nedavno je odr\u017eana i sve\u010dana promocija rada koji je nosio naziv &#8220;Mehanizam inhibicijskog u\u010dinka flavonoida na citokrom P450 3A4&#8221;, pi\u0161e Ve\u010dernji list BiH. 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